background


Product Information:

PCSK9-IN-13

PCSK9-IN-13(compound 3f) is a potent PCSK9 inhibitor, which can antagonize low-density lipoprotein (LDL) receptor binding by binding to PCSK9, with an IC50 of 537 nM.

Cat. No.: EX-A7797    Purity: >98%
Chemical
Chemical structure of PCSK9-IN-13


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
5mg385In-stock
10mg485In-stock
25mg885In-stock
50mgget quoteIn-stock
100mgget quoteIn-stock


CAS No.2244129-23-3
Purity>98%
FormulaC30H33N5O2
Mol Weight495.6153
AppearanceSolid powder
SolubilitySoluble in DMSO
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Benny J. Evison, et al. A small molecule inhibitor of PCSK9 that antagonizes LDL receptor binding via interaction with a cryptic PCSK9 binding groove.Bioorganic & Medicinal Chemistry

Data SheetData sheet of PCSK9-IN-13
CoACoA of PCSK9-IN-13
SDSSDS of PCSK9-IN-13
Smiles:O=C(C1=CC(OC2=CC=CC=C2)=C(C=C1)C)NC3=CC(N4C=C(N=C4)C)=CC(CN5C[C@H](CCC5)N)=C3

KEYWORDS: buy PCSK9-IN-13 | PCSK9-IN-13 supplier | purchase | cost | manufacturer | order | distributor | buy 2244129-23-3 | 2244129-23-3 supplier